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Product Name | SCH 442416 |
Description | A potent, brain-permeable, and selective A2AR antagonist; selective for A2AR over A1R, A2BR, and A3R (Kis = 0.048, 1,111, >10,000, and >10,000 nM, respectively) using human recombinant receptors; selective for A2AR over A1R and A3R in rat cerebral membranes (Kis = 0.50, 1,815, and >10,000 nM, respectively); is taken up preferentially by liver, adrenal gland, kidney, and lungs, and by the striatum in the brain; attenuates adenosine-mediated and A2AR agonist-induced arteriole dilation at a concentration of 10 µM |
Size | 1 mg |
Concentration | n/a |
Applications | n/a |
Other Names | Sch442416 adenosine A2 SCH442416 SCH-442,416 |
Gene, Accession, CAS # | CAS: 316173-57-6 |
Catalog # | 22233-1 |
Price | |
Order / More Info | SCH 442416 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |
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