| 产品详情 |
| Edit |   |
|---|
| Product Name | Carvedilol |
|---|
| Description | A non-selective β-adrenergic receptor antagonist (Kds = 1.78, 0.4, and 5.01 nM for β1-, β2-, and β3-ARs, respectively); also binds to α1-, but not α2-, adrenergic receptors (Kis = 0.81 and 3,400 nM, respectively); reverses increases in heart rate induced by isoproterenol in isolated guinea pig atria (Kb = 0.8 nM); induces relaxation of isolated precontracted guinea pig trachea (Kb = 1.3 nM); prevents epinephrine-induced premature ventricular beats in a rat model of arrhythmia (IC50 = 0.25 mg/kg); inhibits the contractile response to norepinephrine in isolated rabbit aorta (Kb = 11 nM); decreases systolic blood pressure and heart rate in rat models of hypertension at 3-30 mg/kg |
|---|
| Size | 250 mg |
|---|
| Concentration | n/a |
|---|
| Applications | n/a |
|---|
| Other Names | BM 14190 |
|---|
| Gene, Accession, CAS # | CAS: 72956-09-3 |
|---|
| Catalog # | 15418-250 |
|---|
| Price | |
|---|
| Order / More Info | Carvedilol from CAYMAN CHEMICAL COMPANY |
|---|
| Product Specific References | n/a |
|---|
| 产品资料 |
|
|