产品名称 Centrinone B from TOCRIS BIOSCIENCE
产品货号 5690/10
产品价格 现货询价,电话:010-67529703
产品规格 10 mg
产品品牌 TOCRIS BIOSCIENCE
产品概述
产品详情
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Product NameCentrinone B
DescriptionHigh affinity and selective PLK4 inhibitor (Ki = 0.6 nM). Exhibits >2000-fold selectivity for PLK4 over Aurora A and Aurora B. Depletes centriole and centrosome levels in vitro. Induces cell cycle arrest in normal human cell lines in a p53-dependent manner. Purity 98%. MW (observed): 631.67
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names2-[[2-Fluoro-4-[[(2-fluoro-3-nitrophenyl)methyl]sulfonyl]phenyl]thio]-5-methoxy-N-(5-methyl-1H-pyrazol-3-yl)-6-(1-piperidinyl)-4-pyrimidinamine. LCR 323
Gene, Accession, CAS #CAS: 1798871-31-4
Catalog #5690/10
Price
Order / More InfoCentrinone B from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 28811500
产品资料