| 产品详情 |
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| Product Name | EPZ005687 |
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| Description | A potent, selective inhibitor of the lysine methyltranferase EZH2 (Ki = 24 nM), the enzymatic subunit of PRC2; blocks trimethylation of the PRC2 target H3K27 (IC50 = 80 nM), decreasing the proliferation of lymphoma cells carrying mutant, but not wild-type, EZH2 |
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| Size | 50 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | potent selective inhibitors inhibits inhibition epigenetics histones modification modifies lysine methyltransferases cancers EZH2 enzymatic subunits polycomb repressive complex 2 complex-2 complex2 prc2 prc 2 prc-2 substrates S-adenosylmethionine proteins targets EPZ-005687 EPZS 005687 5687 EPZ-5687 EPZ5687 |
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| Gene, Accession, CAS # | CAS: 1396772-26-1 |
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| Catalog # | 13966-50 |
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| Price | |
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| Order / More Info | EPZ005687 from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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