产品名称 JZP 361 from TOCRIS BIOSCIENCE
产品货号 5851/10
产品价格 现货询价,电话:010-67529703
产品规格 10 mg
产品品牌 TOCRIS BIOSCIENCE
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Product NameJZP 361
DescriptionPotent and selective reversible MAGL inhibitor (IC50 = 46 nM). Exhibits 35-fold and 150-fold higher selectivity over human FAAH and ABHD6, respectively (IC50 values are 1.79 and 7.24 μM, respectively). Displays affinity for H1 receptors (pA2 = 6.81). Exhibits no activity at cannabinoid receptors at 10 μM. Purity 99%. MW (observed): 405.88
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names[4-(8-Chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl](1H-1,2,4-triazol-1-yl)methanone
Gene, Accession, CAS #CAS: 1680193-80-9
Catalog #5851/10
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Order / More InfoJZP 361 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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