产品详情 |
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Product Name | GSK 343 |
Description | Potent and selective SAM-competitive EZH2 inhibitor (IC50 = 4 nM). Exhibits >60 fold selectivity for EZH2 over EZH1 and a range of other methyltransferases. Decreases H3K27me3 levels in breast cancer cells in vitro. Inhibits proliferation of prostate cancer cell lines in vitro. Purity 98%. MW (observed): 541.69 |
Size | 50 mg |
Concentration | n/a |
Applications | n/a |
Other Names | N-[(1,2-Dihydro-6-methyl-2-oxo-4-propyl-3-pyridinyl)methyl]-1-(1-methylethyl)-6-[2-(4-methyl-1-piperazinyl)-4-pyridinyl]-1H-indazole-4-carboxamide |
Gene, Accession, CAS # | CAS: 1346704-33-3 |
Catalog # | 6128/50 |
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Order / More Info | GSK 343 from TOCRIS BIOSCIENCE
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Product Specific References | n/a |
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