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Product Name | Fendiline (hydrochloride) |
Description | An α2-adrenergic receptor antagonist (Kd = 2.6 µM) and an L-type calcium channel blocker (IC50 = 17 µM) well-known for its coronary vasodilator effects; inhibits K-Ras plasma membrane localization (IC50 = 9.64 µM), blocking the proliferation of K-Ras-transformed tumor cells |
Size | 5 g |
Concentration | n/a |
Applications | n/a |
Other Names | 119959-32-9 13042-18-7 calcium channel blocker Ca2+ antagonist vasodilation hypertension cardiology signal transduction cancer ion pump biochemical receptor vascular disease Cordan Fendilar Phenoxan Sensit Sensite α2-adrenergic L-type coronary vasodilator inhibit inhibition K-Ras KRas plasma membrane localization tumor |
Gene, Accession, CAS # | CAS: 13636-18-5 |
Catalog # | 17295-5 |
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Order / More Info | Fendiline (hydrochloride) from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |
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