| 产品详情 |
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| Product Name | CPI-637 |
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| Description | An inhibitor of CBP/EP300 bromodomains (IC50s = 30 and 51 nM in a TR-FRET assay); selective for CBP and EP300 over the BET family of bromodomains (IC50s = >10 µM); is active at bromodomain BRD9 (IC50 = 0.73 µM); inhibits CBP (IC50 = 0.3 µM in a BRET assay) and inhibits MYC expression (EC50 = 0.6 µM) in AMO-1 cells |
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| Size | 1 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | CPI637 fluorescence resonance energy transfer cAMP EP-300 TRFRET BRD-9 AMO1 |
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| Gene, Accession, CAS # | CAS: 1884712-47-3 |
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| Catalog # | 23500-1 |
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| Price | |
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| Order / More Info | CPI-637 from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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