产品名称 SR 1664 from CAYMAN CHEMICAL COMPANY
产品货号 11086-5
产品价格 现货询价,电话:010-67529703
产品规格 5 mg
产品品牌 CAYMAN CHEMICAL COMPANY
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Product NameSR 1664
DescriptionA small molecule that blocks phosphorylation of PPARγ by Cdk5 (IC50 = 80 nM; Ki = 28.7 nM) without exhibiting agonist activity at the PPARγ receptor; demonstrates potent, dose-dependent anti-diabetic effects in obese mice without inducing fluid retention and weight gain or inhibiting bone formation
Size5 mg
Concentrationn/a
Applicationsn/a
Other Namesantidiabetics PPARγ inhibitors inhibits inhibitions insulin sensitivity Cdk5 cyclin-dependent kinases 5 diabetes obesity obese metabolic syndromes nuclear receptors peroxisomes proliferator-activated receptors γ g gamma .gamma. PPARg PPARgamma PPAR.gamma. SR1664 SRs 1664 SR-1664 Cdks five potent fluids retention weight gains inhibiting bones formations phosphorylation anti-diabetic
Gene, Accession, CAS #CAS: 1338259-05-4
Catalog #11086-5
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Order / More InfoSR 1664 from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
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