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Product Name | TC ASK 10 |
Description | Potent ASK1 inhibitor (IC50 = 14 nM); displays selectivity for ASK1 over other kinases including ASK2 (IC50 = 0.51 μM), MEKK1, TAK1, IKKβ, ERK1, JNK1, p38α, GSK-3β, PKCθ and B-raf (IC50 values are > 10 μM). Blocks downstream JNK1/p38 phosphorylation in cells. Orally bioavailable. Purity 98%. MW (observed): 432.35 |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 4-(1,1-Dimethylethyl)-N-[6-(1H-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide dihydrochloride |
Gene, Accession, CAS # | CAS: 1005775-56-3 |
Catalog # | 4825/10 |
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Order / More Info | TC ASK 10 from TOCRIS BIOSCIENCE
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Product Specific References | n/a |
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