产品详情 |
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Product Name | VUF 10166 |
Description | High affinity 5-HT3 receptor antagonist (IC50 values are 0.04 and 22 nM for human 5HT3A and 5-HT3AB receptors respectively). Exhibits partial agonist activity at 5-HT3A receptors at higher concentrations (EC50 = 5.2 μM). Also histamine H4 receptor antagonist (pKi = 6.64 in HEK cells). Purity 98%. MW (observed): 262.74 |
Size | 50 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 2-Chloro-3-(4-methyl-1-piperazinyl)quinoxaline |
Gene, Accession, CAS # | CAS: 155584-74-0 |
Catalog # | 4532/50 |
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Order / More Info | VUF 10166 from TOCRIS BIOSCIENCE
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Product Specific References | n/a |
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