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| Product Name | Sumanirole maleate |
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| Description | High affinity D2 receptor agonist (EC50 values are between 17 and 75 nM in cell-based assays). Originally reported to exhibit >200-fold selectivity for the D2 receptor versus other dopamine receptor subtypes (Ki values are 9.0, 1940, >2190 and >7140 for D2, D3, D4 and D1 receptors respectively). More recently reported to be around 32-fold selective for D2 over D3 receptors (Ki values are 17.1 and 546 nM respectively). Exhibits antiParkinsonian activity. Purity 98%. MW (observed): 319.31 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | (R)-5,6-Dihydro-5-(methylamino)-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (2Z)-2-butenedioate |
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| Gene, Accession, CAS # | CAS: 179386-44-8 |
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| Catalog # | 2773/10 |
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| Order / More Info | Sumanirole maleate from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 30175527 |
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| 产品资料 |
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