产品名称 R 1530 from TOCRIS BIOSCIENCE
产品货号 4885/10
产品价格 现货询价,电话:010-67529703
产品规格 10 mg
产品品牌 TOCRIS BIOSCIENCE
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Product NameR 1530
DescriptionMulti-kinase inhibitor. Exhibits inhibitory activity against Chk2, KDR, FGFR, Aurora A kinase and Cdk2 (IC50 values are 24, 34, 50, 58 and 88 nM respectively). Also binds VEGFR-2, FGFR1 and PDGFRβ (Kd values are 0.015, 0.061 and 0.088 μM respectively). Displays antiproliferative activity in vitro; inhibits mitosis and angiogenesis. Orally bioavailable. Purity 98%. MW (observed): 356.78
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names5-(2-Chlorophenyl)-7-fluoro-1,2-dihydro-8-methoxy-3-methylpyrazolo[3,4-b][1,4]benzodiazepine
Gene, Accession, CAS #CAS: 882531-87-5
Catalog #4885/10
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Order / More InfoR 1530 from TOCRIS BIOSCIENCE
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