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| Product Name | GR 159897 |
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| Description | A potent, selective, non-peptide, orally active neurokinin NK2 receptor antagonist. Competes for binding of [3H]GR100679 to hNK2-transfected CHO cells with a pKi of 9.5. Inhibits NK2 receptor-mediated contraction of guinea pig trachea with a pA2 of 8.7. Anxiolytic in vivo. Purity 97%. MW (observed): 414.54 |
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| Size | 50 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 5-Fluoro-3-[2-[4-methoxy-4-[[(R)-phenylsulphinyl]methyl]-1-piperidinyl]ethyl]-1H-indole |
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| Gene, Accession, CAS # | CAS: 158848-32-9 |
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| Catalog # | 1274/50 |
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| Price | |
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| Order / More Info | GR 159897 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 21188216, 21368235, 22363709, 22758653 |
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