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| Product Name | Conivaptan (hydrochloride) |
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| Description | A vasopressin V1A and V2 receptor antagonist (Kis = 0.48 and 3.04 nM for rat liver V1A and kidney V2, respectively); competitively inhibits oxytocin binding to rat uterine oxytocin receptors (Ki = 44 nM) but has no effect on AVP binding to anterior pituitary V1B receptors at concentrations up to 100 µM in a radioligand binding assay; suppresses AVP-induced increases in intracellular calcium in VSMCs and the pressor response in pithed rats; increases urine output and decreases urine osmolality in dehydrated conscious rats in a dose-dependent manner; reduces brain edema and blood-brain barrier disruption in a mouse experimental stroke model, |
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| Size | 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | YM-087 |
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| Gene, Accession, CAS # | CAS: 168626-94-6 |
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| Catalog # | 23728-5 |
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| Order / More Info | Conivaptan (hydrochloride) from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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