产品名称 Saxagliptin (hydrochloride) from CAYMAN CHEMICAL COMPANY
产品货号 23697-1
产品价格 现货询价,电话:010-67529703
产品规格 1 mg
产品品牌 CAYMAN CHEMICAL COMPANY
产品概述
产品详情
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Product NameSaxagliptin (hydrochloride)
DescriptionA potent DPP-4 inhibitor (Ki = 0.6 nM); inhibits DPP-4 ex vivo (ED50 = 0.12 µmol/kg) in plasma from normal fasted rats; reduces plasma glucose levels in Zuckerfa/fa diabetic rats in a dose-dependent manner when administered orally in doses ranging from 0.3-3 mg/kg; increases plasma insulin levels and improves glucose clearance in ob/ob mice; induces systolic and diastolic dysfunction, reduces contractile force, and exacerbates ischemia-reperfusion injury-induced cardiac dysfunction in isolated guinea pig hearts
Size1 mg
Concentrationn/a
Applicationsn/a
Other NamesBMS-477118
Gene, Accession, CAS #CAS: 709031-78-7
Catalog #23697-1
Price
Order / More InfoSaxagliptin (hydrochloride) from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
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