产品名称 Valdecoxib - SC 65872 | Bextra
产品货号 Axon 2106 CAS [181695-72-7] MF C16H14N2O3SMW 314.36 Purity: 99% Soluble in DMSO Description NSAID. Highly selective and potent inhibitor of COX-2 in human whole blood and against the recombinant human enzyme, showing exceptional potency after oral administration. Valdecoxib showed weak inhibitory activity against COX-1 (IC50 = 140 µM), and potent activity against COX-2 (IC50 = 0.005 µM) References Certificates Categories Extra info JJ Talley et al. 4-[5-Methyl-3-phenylisoxazol-4-yl]- benzenesulfonamide, valdecoxib: a potent and selective inhibitor of COX-2. J. Med. Chem. 2000, 43(5), 775-777.  Certificate of Analysis Material Safety Data Sheet CNS Immunology Pain & Inflammation EC 1.14.99.1 COX Pfizer Licensed Products Selecive COX-2 inhibitor Chemical name 4-(5-methyl-3-phenylisoxazol-4-yl)benzenesulfonamide Source information Pfizer compound; Sold for research purposes under agreement from Pfizer Inc. Parent CAS No. [181695-72-7] Order Size Unit Price Stock 10 mg €80.00 In Stock
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Valdecoxib - SC 65872 | Bextra

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 2106

CAS [181695-72-7]

MF C16H14N2O3S
MW 314.36

  • Purity: 99%
  • Soluble in DMSO

Valdecoxib

Description

NSAID. Highly selective and potent inhibitor of COX-2 in human whole blood and against the recombinant human enzyme, showing exceptional potency after oral administration. Valdecoxib showed weak inhibitory activity against COX-1 (IC50 = 140 µM), and potent activity against COX-2 (IC50 = 0.005 µM)
Selecive COX-2 inhibitor

Chemical name

4-(5-methyl-3-phenylisoxazol-4-yl)benzenesulfonamide

Source information

Pfizer compound; Sold for research purposes under agreement from Pfizer Inc.

Parent CAS No.

[181695-72-7]

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