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产品名称 PF 04981517 - CYP3cide | PF 4981517
产品货号 Axon 2026 CAS [1390637-82-7] MF C26H32N8MW 456.59 Purity: 98% Optical purity: Optically pure Soluble in 0.1N HCl(aq) and DMSO Description Potent and selective inhibitor of Cytochrome P450 3A4 (CYP3A4) with IC50 value of 30 nM; inactivates human CYP3A4 in an efficient and time-dependent manner References Certificates Categories Extra info RL Walksky et al. Selective mechanism-based inactivation of CYP3A4 by CYP3cide (PF-04981517) and its utility as an in vitro tool for delineating the relative roles of CYP3A4 versus CYP3A5 in (...). Drug Metab. Dispos. 2012, 40(9), 1686-1697.    Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology Diabetes & Metabolism EC 1.14.13.97 Cytochrome P450 Pfizer Licensed Products Inhibitor of Cytochrome P450 3A4 (CYP3A4) Chemical name (S)-1-methyl-3-(1-methyl-5-p-tolyl-1H-pyrazol-4-yl)-4-(3-(piperidin-1-yl)pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine Source information Pfizer compound; Sold for research purposes under agreement from Pfizer Inc. Parent CAS No. [1390637-82-7] Order Size Unit Price Stock 10 mg €110.00 In Stock
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产品品牌 axonmedchem
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PF 04981517 - CYP3cide | PF 4981517

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 2026

CAS [1390637-82-7]

MF C26H32N8
MW 456.59

  • Purity: 98%
  • Optical purity: Optically pure
  • Soluble in 0.1N HCl(aq) and DMSO

PF 04981517

Description

Potent and selective inhibitor of Cytochrome P450 3A4 (CYP3A4) with IC50 value of 30 nM; inactivates human CYP3A4 in an efficient and time-dependent manner
Inhibitor of Cytochrome P450 3A4 (CYP3A4)

Chemical name

(S)-1-methyl-3-(1-methyl-5-p-tolyl-1H-pyrazol-4-yl)-4-(3-(piperidin-1-yl)pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine

Source information

Pfizer compound; Sold for research purposes under agreement from Pfizer Inc.

Parent CAS No.

[1390637-82-7]
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