产品名称 WAY 100635 maleate
产品货号 Axon 2424 CAS [1092679-51-0] MF C25H34N4O2.C4H4O4MW 538.64 Purity: 98% Soluble in water and DMSO Description Prototypical 5-HT1A receptor antagonist with D4 agonist activity (Ki values 2.2 nM, 6260 nM, 24 nM, >10,000 nM, 20 nM, 322 nM, and 16 nM for 5-HT1A, 5-HT2A, 5-HT2B, 5-HT7, α1A, α1B, and D4, respectively). The HCl salt of WAY 100635 is available as well (Axon 1086) References Certificates Categories Extra info B.R. Chemel et al. WAY-100635 is a potent dopamine D4 receptor agonist. Psychopharmacology (Berl). 2006 Oct;188(2):244-51.   EA Forster et al. A pharmacological profile of the selective silent 5-HT1A receptor antagonist WAY-100635. Eur. J. Pharmacol. 1995, 281, 81-88.    F. Mangin et al. Moderate chemical modifications of WAY-100635 improve the selectivity for 5-HT1A versus D4 receptors. Bioorg Med Chem Lett. 2012 Jul 15;22(14):4550-4. Certificate of Analysis Material Safety Data Sheet Cell Signaling & Oncology CNS 5-HT1A D4 Adrenoceptor α1 A19 5-HT1A antagonist with D4 agonistic properties Chemical name Cyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide maleate Parent CAS No. [162760-96-5] Order Size Unit Price Stock 10 mg €125.00 In Stock
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WAY 100635 maleate

Based on 8 reference(s) in Google Scholar 9 10 8

Axon 2424

CAS [1092679-51-0]

MF C25H34N4O2.C4H4O4
MW 538.64

  • Purity: 98%
  • Soluble in water and DMSO

WAY 100635 maleate

Description

Prototypical 5-HT1A receptor antagonist with D4 agonist activity (Ki values 2.2 nM, 6260 nM, 24 nM, >10,000 nM, 20 nM, 322 nM, and 16 nM for 5-HT1A, 5-HT2A, 5-HT2B, 5-HT7, α1A, α1B, and D4, respectively).

The HCl salt of WAY 100635 is available as well (Axon 1086)

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