| 产品详情 |
| Edit |   |
|---|
| Product Name | SCH 442416 |
|---|
| Description | A potent, brain-permeable, and selective A2AR antagonist; selective for A2AR over A1R, A2BR, and A3R (Kis = 0.048, 1,111, >10,000, and >10,000 nM, respectively) using human recombinant receptors; selective for A2AR over A1R and A3R in rat cerebral membranes (Kis = 0.50, 1,815, and >10,000 nM, respectively); is taken up preferentially by liver, adrenal gland, kidney, and lungs, and by the striatum in the brain; attenuates adenosine-mediated and A2AR agonist-induced arteriole dilation at a concentration of 10 µM |
|---|
| Size | 10 mg |
|---|
| Concentration | n/a |
|---|
| Applications | n/a |
|---|
| Other Names | Sch442416 adenosine A2 SCH442416 SCH-442,416 |
|---|
| Gene, Accession, CAS # | CAS: 316173-57-6 |
|---|
| Catalog # | 22233-10 |
|---|
| Price | |
|---|
| Order / More Info | SCH 442416 from CAYMAN CHEMICAL COMPANY |
|---|
| Product Specific References | n/a |
|---|
| 产品资料 |
|
|