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Product Name | Zosuquidar trihydrochloride |
Description | Purity >98% by HPLC. Zosuquidar is a potent P-glycoprotein (P-gp) inhibitor (Kd = 79 nM). Zosuquidar binds with high affinity to P-glycoprotein and inhibits P-glycoprotein-mediated multidrug resistance (MDR). Restores doxorubicin sensitivity in P-gp-expressing multidrug (MDR) resistant cancer cell lines. |
Size | n/a |
Concentration | n/a |
Applications | n/a |
Other Names | (AR)-4-[(1aA,6A,10bA)-1,1-Difluoro-1,1a,6,10b-tetrahydrodibenzo[a,e]cyclopropa[c]cyclohepten-6-yl]-A-[(5-quinolinyloxy)methyl]-1-piperazineethanol trihydrochloride, LY335979 |
Gene, Accession, CAS # | CAS: 167465-36-3 |
Catalog # | LS-H3537 |
Price | |
Order / More Info | Zosuquidar trihydrochloride from LIFESPAN BIOSCIENCES INC. |
Product Specific References | n/a |
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