| 产品详情 |
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| Product Name | PFI-2 |
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| Description | MW: 499.52. Purity ≥98% by HPLC. PFI-2 is a novel potent and selective SETD7 histone lysine methyltransferase inhibitor (IC50 ~2 nM). It has > 100-fold selectivity over other methyltransferases and other non-epigenetic targets. PFI-2 has been shown to bind to SETD7 by ITC (Kd = 18 nM); and biotinylated PFI-2 interacts with SETD7 in pull-down studies. |
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| Size | 5 mg, 25 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | [(R)-8-fluoro-N- (1-oxo-1- (pyrrolidin-1-yl)-3- (3- (trifluoromethyl) phenyl) propan-2-yl)-1; 2; 3; 4-tetrahydroisoquinoline-6-sulfonamide] |
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| Gene, Accession, CAS # | CAS: 1627676-59-8 |
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| Catalog # | MBS846401 |
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| Order / More Info | PFI-2 from MYBIOSOURCE INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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