| 产品名称 | Pimobendan - Inhibitors / Activators - Phosphodiesterase(s) |
| 产品货号 | 27638-1 |
| 产品价格 | 现货询价，电话：010-67529703 |
| 产品规格 | 10 mg |
| 产品品牌 | bpsbioscience |
| 产品概述 | |
| 产品详情 |
MW: 334.37 Da
CAS Registry #: 74150-27-9
Formula: C19H18N4O2
Target: PDE3
Description: Pimobendan is a selective inhibitor of PDE3 with IC50 of 0.32 µM.
Synonym(s): pimobendane; 3-[2-(4-methoxyphenyl)-3H-benzimidazol-5-yl]-4-methyl-4,5-dihydro-1H-pyridazin-6-one
Biological Activity: Pimobendan exhibits selective inhibition of PDE III isolated from guinea pig cardiac muscle with IC50 of 0.32 uM compared to the inhibition of PDE I and PDE II (IC50s>30 µM). Pimobendan inhibits the activity of cAMP-PDE III with IC50 of 2.4 µM.
Storage / Stability: Store at or below –20°C. Solid form is stable at least 12 months from date of receipt, when stored as directed. Do not store aqueous solutions for more than one day. Reference(s): Boyle KL, Leech E. J Vet Emerg Crit Care (San Antonio). 2012 Aug;22(4):398-408.
Scientific Category: PDE Inhibitor
Product Type: Inhibitor
Data shown is lot-specific. Contact us for specific information on other lots.
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